Compile Data Set for Download or QSAR
Found 5 from The Burnham Institute
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Burnham Institute

LigandPNGBDBM15186(4-(5-{[(5E)-2-amino-3,7-dicyano-4,6-dimethyl-5H-cy...)copy SMILEScopy InChI
Affinity DataKi:  1.10E+3nM ΔG°:  -8.12kcal/mole IC50: 2.60E+3nMpH: 7.5 T: 2°CAssay Description:The Z-LYTE assay (Invitrogen Corporation) employs a FRET-based, coupled-enzyme format and is based on the differential sensitivity of phosphorylated ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD1W4ZPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Burnham Institute

LigandPNGBDBM15187(3-[(2E)-3-(1H-1,3-benzodiazol-2-yl)prop-2-enoyl]-6...)copy SMILEScopy InChI
Affinity DataKi:  3.90E+3nM ΔG°:  -7.37kcal/mole IC50: 4.50E+3nMpH: 7.5 T: 2°CAssay Description:The Z-LYTE assay (Invitrogen Corporation) employs a FRET-based, coupled-enzyme format and is based on the differential sensitivity of phosphorylated ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD1W4ZPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Burnham Institute

LigandPNGBDBM15188(5-{5-[(1,3-dioxo-2,3-dihydro-1H-inden-2-ylidene)me...)copy SMILEScopy InChI
Affinity DataKi:  2.08E+4nM ΔG°:  -6.38kcal/mole IC50: 2.51E+4nMpH: 7.5 T: 2°CAssay Description:The Z-LYTE assay (Invitrogen Corporation) employs a FRET-based, coupled-enzyme format and is based on the differential sensitivity of phosphorylated ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD1W4ZPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Burnham Institute

LigandPNGBDBM15190(3-(5-{[(5E)-2-amino-3,7-dicyano-4,6-dimethyl-5H-cy...)copy SMILEScopy InChI
Affinity DataIC50: 6.02E+4nMpH: 7.5 T: 2°CAssay Description:The Z-LYTE assay (Invitrogen Corporation) employs a FRET-based, coupled-enzyme format and is based on the differential sensitivity of phosphorylated ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD1W4ZPubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
The Burnham Institute

LigandPNGBDBM15189(4-(5-{[(5E)-2-amino-3,7-dicyano-4,6-dimethyl-5H-cy...)copy SMILEScopy InChI
Affinity DataIC50: 1.26E+5nMpH: 7.5 T: 2°CAssay Description:The Z-LYTE assay (Invitrogen Corporation) employs a FRET-based, coupled-enzyme format and is based on the differential sensitivity of phosphorylated ...More data for this Ligand-Target Pair
In DepthDetails Article
BindingDB Entry DOI: 10.7270/Q2KD1W4ZPubMed